Sat. Oct 26th, 2024

5-CT Maleate

5-CT MaleateBand: www.medchemexpress.comAgonist at 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5 and 5-HT7 serotonin receptorsCAS No: 74885-72-6   Chemical Name: 5-Carboxamidotryptamine maleate salt (+)-JQ-2 Molecular Formula C15H17N3O5 Molecular Weight 319.31 CAS Numbers 74885-72-6 Storage Condition…

A-412997 Dihydrochloride

A-412997 DihydrochlorideBand: www.medchemexpress.comSelective agonist of dopamine D4 receptorCAS No: 630116-49-3   Chemical Name: N-(3-Methylphenyl)-4-(2-pyridinyl)-1-piperidineacetamide Dihydrochloride Rigosertib (sodium) Molecular Formula C19H25Cl2N3O Molecular Weight 382.33 CAS Numbers 630116-49-3 Storage Condition 0°C (short term), -20°C…

77-LH-28-1 Oxalate

77-LH-28-1 OxalateBand: www.medchemexpress.comCNS penetrant, selective M1 muscarinic receptor agonistCAS No:  560085-12-3, 560085-11-2(Free Base)   Chemical Name: 1--3,4-dihydroquinolin-2-one Oxalate PF-2545920 Molecular Formula 560085-12-3 and 560085-11-2 (Free Base) Molecular Weight C23H34N2O5 CAS Numbers 418.53…

4P-PDOT

4P-PDOTBand: www.medchemexpress.comSelective antagonist of melatonin receptor subtype 2 (MT2)CAS No: 134865-74-0   Chemical Name: 4-P-PDOT; 4PPDOT; AH-024; (+/-)-cis-N-(4-phenyl-1,2,3,4-tetrahydronaphthalen-2-yl)propanamide SCR7 Molecular Formula C19H21NO Molecular Weight 279.38 CAS Numbers 134865-74-0 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18493315

(S)-PD-126055 (EMA401)

(S)-PD-126055 (EMA401)Band: www.medchemexpress.comMore active S-enantiomer of EMA400 (AOB4655), a potent and highly selective AT2R antagonist CAS No: 1316755-16-4   Chemical Name: (S)-5-Benzyloxy-2-diphenylacetyl-6-methoxy-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid ARRY-520 Molecular Formula C32H29NO5 Molecular Weight 507.58 CAS…

(S)-FTY720P

(S)-FTY720PBand: www.medchemexpress.comA sphingosine 1-phosphate (S1PR) receptor agonist CAS No:402616-26-6 CP-673451 Molecular Formula C19H34NO5P Molecular Weight 387.45 CAS Numbers 402616-26-6 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Stock…

Yohimbine hydrochloride

Yohimbine hydrochlorideBand: www.medchemexpress.comPotent antagonist of alpha2-adrenergic receptor, showing moderate affinity for the alpha1 receptor, 5-HT1A, 5-HT1B, 5-HT1D, 5-HT1F, 5-HT2B, and D2 receptors, and weak affinity for the 5-HT1E, 5-HT2A, 5-HT5A,…

Kv2-IN-A1

Kv2-IN-A1Band: www.medchemexpress.comNovel Kv2.1 and Kv2.2 inhibitor  CAS No: 689297-68-5   Chemical Name: 3-(3-Chlorophenyl)-N-butyramide SAR405838 Molecular Formula C20H17ClN4OS Molecular Weight 396.89 CAS Numbers 689297-68-5 Storage Condition 0°C (short term), -20°C (long term), desiccated…

HUP30

HUP30Band: www.medchemexpress.comNovel vasorelaxing agent, stimulating soluble guanylyl cyclase, activating K+ channels, and blocking extracellular Ca2+ influxCAS No: 312747-21-0   Chemical Name: N-(6-Nitro-2-benzothiazolyl)-cyclohexanecarboxamide GANT 61 Molecular Formula C14H15N3O3S Molecular Weight 305.35 CAS Numbers…

Glybenclamide

GlybenclamideBand: www.medchemexpress.comNLRP3 inhibitor, selectively blocking ATP-sensitive K+ channels; high affinity binding sites found in brain, pancreatic β cells, and cardiovascular systemCAS No: 10238-21-8   Chemical Name: 5-​Chloro-​N-​​-​2-​methoxybenzamide, Glyburide, N-p-​​benzenesulfonyl-​N′-cyclohexylurea AZD-8055 Molecular Formula…