Sat. Oct 26th, 2024

CID-85469571

CID-85469571Band: www.medchemexpress.comThe first selective antagonist of orphan receptor GPR18 Olcegepant Molecular Formula C120H17ClN2O2S Molecular Weight 384.88 CAS Numbers 1627710-30-8 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO…

CID-16020046

CID-16020046Band: www.medchemexpress.comSelective GPR55 antagonistCAS No: 834903-43-4 Chemical Name: 4-pyrazol-5-yl]benzoic acid; 4-pyrazol-5(1H)-yl]-benzoic acid Bafetinib Molecular Formula C25H19N3O4 Molecular Weight 425.44 CAS Numbers 834903-43-4 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18496505

APD668

APD668Band: www.medchemexpress.comNovel agonist of the orphan G-protein coupled receptor GPR119CAS No: 832714-46-2   Chemical Name: JNJ-28630368; Propan-2-yl 4-pyrimidin-4-yl]oxypiperidine-1-carboxylate Volasertib Molecular Formula C21H24FN5O5S Molecular Weight 477.51 CAS Numbers 832714-46-2 Storage Condition 0°C (short…

APD597

APD597Band: www.medchemexpress.comSecond generation agonist of the orphan G-protein coupled receptor GPR119 CAS No: 897732-93-3   Chemical Name: JNJ-38431055; Propan-2-yl 4-pyrimidin-4-yl]oxypiperidine-1-carboxylate Azeliragon Molecular Formula C21H29N5O6S Molecular Weight 479.552 CAS Numbers 897732-93-3 Storage Condition…

PD-34799-SA

PD-34799-SABand: www.medchemexpress.comInhibitor of the orexin type 1 receptorCAS No:1021-11-0 Chemical Name: N-​(6,8-​Difluoro-​2-​methyl-​4-​quinolinyl)​-​N′-urea (-)-DHMEQ Molecular Formula C19H18F2N4O Molecular Weight 356.37 CAS Numbers 288150-92-5 Storage Condition 0°C (short term), -20°C (long term), desiccated…

MK-4305

MK-4305Band: www.medchemexpress.comA dual orexin receptor antagonist that blocks both OX1R and OX2R CAS No:1030377-33-3 PCI-32766 Molecular Formula C23H23ClN6O2 Molecular Weight 450.9 CAS Numbers 1030377-33-3 Storage Condition 0°C (short term), -20°C (long…

MK-3697

MK-3697Band: www.medchemexpress.comAn isonicotinamide small molecule, acting as a potent and selective Orexin receptor antagonistCAS No:1224846-01-8 Calicheamicin Molecular Formula C23H21N5O3S Molecular Weight 447.5 CAS Numbers 1224846-01-8 Storage Condition 0°C (short term),…

MDK5220 (Orexin 2 Receptor Agonist)

MDK5220 (Orexin 2 Receptor Agonist)Band: www.medchemexpress.comNovel potent and selective Orexin2 receptor agonist CAS No: 1796565-52-0 Chemical Name: 4-Methoxy-N,N-dimethyl-3-(N-(3-((2-(3-methylbenzamido)ethyl)amino)phenyl)sulfamoyl)--3-carboxamide Brigatinib Molecular Formula C32H34N4O5S Molecular Weight 586.707 CAS Numbers 1796565-52-0 Storage Condition 0°C…

Almorexant HCl

Almorexant HClBand: www.medchemexpress.coma dual antagonist of the orexin 1 and 2 receptorsCAS No:913358-93-7 UNC0639 Molecular Formula C29H32ClF3N2O3 Molecular Weight 549.02 CAS Numbers 913358-93-7 Storage Condition 0°C (short term), -20°C (long…

Almorexant

AlmorexantBand: www.medchemexpress.comA potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.CAS No:871224-64-5 FK867 Molecular…