BarbadinBand: www.medchemexpress.comNovel selective β-arrestin/β2-adaptin inhibitor, blocking agonist-promoted endocytosis of the prototypical β2-adrenergic (β2AR), V2-vasopressin (V2R) and angiotensin-II type-1 (AT1R) receptors, showing no affectinng on β-arrestin-independent (transferrin) or AP2-independent (endothelin-A) receptor…
CMF-019 PotassiumBand: www.medchemexpress.comThe first potent biased small molecule agonist at the apelin receptor, increasing cardiac contractility in vivoCAS No: 1993426-69-9 Chemical Name: Potassium 3(S)-{-amino}-5-methyl-hexanoate LCL162 Molecular Formula C25H32KN3O3S Molecular Weight 493.70…
CMF-019Band: www.medchemexpress.comThe first potent biased small molecule agonist at the apelin receptor, increasing cardiac contractility in vivoCAS No: 1586787-08-7 Chemical Name: 3(S)-{-amino}-5-methyl-hexanoate TGR-1203 Molecular Formula C25H33N3O3S Molecular Weight 454.60 CAS…
MRT-10Band: www.medchemexpress.comSmoothened (Smo) receptor antagonistCAS No:330829-30-6 Chemical Name: N-amino]thioxomethyl]-3,4,5-trimethoxybenzamide Losmapimod Molecular Formula C24H23N3O5S Molecular Weight 465.52 CAS Numbers 330829-30-6 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…
Rilmenidine hemifumarateBand: www.medchemexpress.comSelective I1 imidazoline receptor agonistCAS No: 207572-68-7 Chemical Name: Oxaminozoline hemifumarate; N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt Paritaprevir Molecular Formula C12H13N2O3 Molecular Weight 238.28 CAS Numbers 207572-68-7 Storage Condition 0°C (short term), -20°C…
ML314Band: www.medchemexpress.comNovel agonist of Neurotesin 1 Receptor (NTR1)CAS No: 1448895-09-7 Chemical Name: 2-Cyclopropyl-6,7-dimethoxy-4-quinazoline THZ2 Molecular Formula C22H26Cl2N2O9 Molecular Weight 421.36 CAS Numbers 858474-14-3 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18497484
JNJ-17203212Band: www.medchemexpress.comPotent TRPV1 (VR1) vanilloid receptor antagonist CAS No: 821768-06-3 Chemical Name: 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic acid (5-trifluoromethylpyridin-2-yl)amide; JNJ17203212 AZD3966 Molecular Formula C17H15F6N5O Molecular Weight 419.32 CAS Numbers 821768-06-3 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18497261
GSK2193874Band: www.medchemexpress.comSelective and orally active blocker of transient receptor potential vanilloid 4 (TRPV4)CAS No: 1336960-13-4 Chemical Name: 3-(-1-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2--4-quinolinecarboxami NVP-BGJ399 Molecular Formula C37H38BrF3N4O Molecular Weight 691.62 CAS Numbers 1336960-13-4 Storage Condition 0°C…
GSK205Band: www.medchemexpress.comSelective Transient receptor potential vanilloid 4 (TRPV4) antagonistCAS No: 1263130-79-5 Chemical Name: N-ethyl]phenyl]-5-(3-pyridinyl)-2-thiazolamine PF-04449914 Molecular Formula C24H24N4S Molecular Weight 400.54 CAS Numbers 1263130-79-5 Storage Condition 0°C (short term), -20°C (long…
AMG-9810Band: www.medchemexpress.comA potent non-vanilloid antagonist of the TRPV1 receptor CAS No: 545395-94-6 Chemical Name: 2E-N-(2,3-Dihydro-1,4-benzodioxin-6-yl)-3--2-Propenamide 4-Deazaneplanocin A (hydrochloride) Molecular Formula C21H23NO3 Molecular Weight 337.4 CAS Numbers 545395-94-6 Storage Condition 0°C (short…