Fri. Oct 18th, 2024

Thiazovivin

ThiazovivinBand: www.medchemexpress.comNovel ROCK inhibitor, enhancing embryonic stem cell (ESCs) survival via ROCK PathwayCAS No: 1226056-71-8   Chemical Name: TZV; N-Benzyl-2-(pyrimidin-4-ylamino)-1,3-thiazole-4-carboxamide TAK-244 Molecular Formula C15H13N5OS Molecular Weight 311.36 CAS Numbers 1226056-71-8 Storage Condition…

SB-431542

SB-431542Band: www.medchemexpress.comInhibitor of the TGF-beta type I receptor kinase activityCAS No: 301836-41-9   Chemical Name: SB431542; 4-(4-(Benzodioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide BYL-721 Molecular Formula C22H16N4O3 Molecular Weight 384.4 CAS Numbers 301836-41-9 Storage Condition 0°C (short term),…

PD 0325901

PD 0325901Band: www.medchemexpress.comA potent and highly selective small molecule MEK (MAPK/ERK Kinase) inhibitorCAS No:391210-10-9 LY2835221 Molecular Formula C16H14F3IN2O4 Molecular Weight 482.19 CAS Numbers 391210-10-9 Storage Condition 0°C (short term), -20°C…

Forskolin

ForskolinBand: www.medchemexpress.comActivator of adenylyl cyclase, possessing anti-hypertensive, positive inotropic, and inhibiting MAP kinaseCAS No: 66575-29-9   Chemical Name: Colforsin; Coleonol; Boforsin; Colforsina; chromen-5-yl] acetate Monomethyl auristatin E Molecular Formula C22H34O7 Molecular Weight…

EPZ004777

EPZ004777Band: www.medchemexpress.comPotent DOT1L Inhibitor; The first-in-class SAM-competitive and selective histone methyl transferase inhibitorChemical Name: 7-amino]carbonyl]amino]propyl](1-methylethyl)amino]-β-D-ribofuranosyl]-7H-pyrrolopyrimidin-4-amine; CAS No: 1338466-77-5 EPZ015668 Molecular Formula C28H41N7O4 Molecular Weight 539.67 CAS Numbers 1338466-77-5 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18502103

CHIR-99021

CHIR-99021Band: www.medchemexpress.comCell-permeable, potent, ATP-competitive, and highly selective GSK-3 inhibitorCAS No: 252917-06-9   Chemical Name: 6-(2-(4-(2,4-Dichlorophenyl)-5-(4-methyl-1H-imidazol-2-yl)-pyrimidin-2-ylamino)ethylamino)-nicotinonitrile PKC414 Molecular Formula C22H18Cl2N8 Molecular Weight 465.34 CAS Numbers 252917-06-9 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18502066

BIX-01294 trihydrochloride

BIX-01294 trihydrochlorideBand: www.medchemexpress.comSelective inhibitor of G9a histone methyltransferase CAS No : 1392399-03-9   Chemical Name: 2-(Hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6,7-dimethoxy-N--4-quinazolinamine trihydrochloride (+)-JQ-3 Molecular Formula C28H38N6O2.3HCl Molecular Weight 600.02 CAS Numbers 1392399-03-9 Storage Condition 0°C (short term), -20°C…

AM580 (NSC 608001, Ro 40-6055)

AM580 (NSC 608001, Ro 40-6055)Band: www.medchemexpress.comSelective RARa agonistCAS No: 102121-60-8   Chemical Name: CD336; 4-benzoic acid Rigosertib (sodium) Molecular Formula C22H25NO3 Molecular Weight 351.4 CAS Numbers 102121-60-8 Storage Condition 0°C (short…

NSC109555 Dimesylate

NSC109555 DimesylateBand: www.medchemexpress.comSelective, reversible, ATP-competitive inhibitorCAS No: 15427-93-7 Chemical Name: DDUG diMS; NCI-C04808; 4,4-Diacetyldiphenylurea bis(guanylhydrazone) bismethanesulfonate PF-2545921 Molecular Formula C21H32N10O7S2 Molecular Weight 600.67 CAS Numbers 15427-93-7 References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/18502001

Hydralazine Hydrochloride

Hydralazine HydrochlorideBand: www.medchemexpress.comInhibits DNA methyltransferase and modulates epigenetic regulation of gene expression. Non-selective MAO-A/B inhibitor; antihypertensive; semicarbazide-sensitive amine oxidase inhibitor.CAS No:304-20-1 SCR8 Molecular Formula C8H8N4 · HCl Molecular Weight 196.64…