IWP-3Band: www.medchemexpress.comAn inhibitor of Wnt production that impairs Wnt pathway activity in vitro with an IC50 value of 40 nMCAS No: 687561-60-0 Chemical Name: 2-pyrimidin-2-yl]thio]-N-(6-methyl-2-benzothiazolyl)-acetamide CHIR-99029 Molecular Formula C22H17FN4O2S3 Molecular Weight 484.6 CAS Numbers…
I-BET151 (GSK1210151A)Band: www.medchemexpress.comSelective BET inhibitorCAS No: 1300031-49-5 Chemical Name: 7-(3,5-Dimethyl-4-isoxazolyl)-1,3-dihydro-8-methoxy-1--2H-imidazoquinolin-2-one hydrochloride; GSK1210151A AT9291 Molecular Formula C23H21N5O3 Molecular Weight 415.44 CAS Numbers 1300031-49-5 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…
HAT Inhibitor IIBand: www.medchemexpress.comNovel p300/CBP-selective histone acetyltransferase inhibitor JIB-12 Molecular Formula C20H16Br2O3 Molecular Weight 464.15 CAS Numbers 932749-62-7 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility DMSO Purity…
GSK682753ABand: www.medchemexpress.comNovel antagonist of oxysterol-induced Epstein–Barr virus induced gene 2 (EBI2) activation CAS No: 1334294-76-6 Chemical Name: 8--3--1-oxa-3,8-diazaspirodecan-2-one Forodesine (hydrochloride) Molecular Formula C23H21Cl3N2O3 Molecular Weight 479.78 CAS Numbers 1334294-76-6 Storage Condition…
GSK3787Band: www.medchemexpress.comPotent and selective peroxisome proliferator-activated receptor δ (PPARδ) antagonist CAS No:188591-46-0 Octreotide (acetate) Molecular Formula C15H12ClF3N2O3S Molecular Weight 392.78 CAS Numbers 188591-46-0 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…
GSK126Band: www.medchemexpress.comPotent, highly selective, S-adenosyl-methionine-competitive, inhibitor of EZH2 methyltransferase activityCAS No: 1346574-57-9 SP2517 Molecular Formula C31H38N6O2 Molecular Weight 526.67 CAS Numbers 1346574-57-9 Storage Condition -20°C 2 years References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/18559251
GSK-J4Band: www.medchemexpress.comHistone demethylase JMJD3/UTX inhibitorCAS No: 1373423-53-0 Chemical Name: N--β-alanine ethyl ester MG-140 Molecular Formula C24H27N5O2 Molecular Weight 417.5 CAS Numbers 1373423-53-0 Storage Condition 0°C (short term), -20°C (long term),…
GSK-J1Band: www.medchemexpress.comPotent and selective inhibitor of the H3K27 histone demethylases JMJD3 and UTXCAS No: 1373422-53-7 Chemical Name: N--β-alanine Deforolimus Molecular Formula C22H23N5O2 Molecular Weight 389.45 CAS Numbers 1373422-53-7 Storage Condition 0°C…
GNE-140 racemicBand: www.medchemexpress.comNovel potent lactate dehydrogenase (LDHA) inhibitor CAS No: 1809794-70-4 Chemical Name: 3-((2-Chlorophenyl)thio)-4-hydroxy-6-(4-morpholinophenyl)-6-(thiophen-3-yl)-5,6-dihydropyridin-2(1H)-one Birinapant Molecular Formula C₂₅H₂₃ClN₂O₃S₂ Molecular Weight 499.04 CAS Numbers 1802977-61-2 Storage Condition 0°C (short term), -20°C (long…
GNE 477Band: www.medchemexpress.comA potent and efficacious dual PI3K/mTOR inhibitorCAS No:1032754-81-6 c-Kit-IN-9 Molecular Formula C21H28N8O3S2 Molecular Weight 504.63 CAS Numbers 1032754-81-6 Storage Condition 0°C (short term), -20°C (long term), desiccated Solubility…